ATX inhibitor 1

CAS No. 2225892-70-4

ATX inhibitor 1 ( —— )

Catalog No. M22925 CAS No. 2225892-70-4

ATX inhibitor 1 is a potent ATX inhibitor (IC50: 1.23 nM, FS-3 and 2.18 nM, bis-pNPP).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 106 Get Quote
5MG 177 Get Quote
10MG 281 Get Quote
25MG 473 Get Quote
50MG 683 Get Quote
100MG 963 Get Quote
200MG Get Quote Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    ATX inhibitor 1
  • Note
    Research use only, not for human use.
  • Brief Description
    ATX inhibitor 1 is a potent ATX inhibitor (IC50: 1.23 nM, FS-3 and 2.18 nM, bis-pNPP).
  • Description
    ATX inhibitor 1 is a potent ATX inhibitor (IC50: 1.23 nM, FS-3 and 2.18 nM, bis-pNPP).
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    PDE
  • Recptor
    ATX
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2225892-70-4
  • Formula Weight
    501.3
  • Molecular Formula
    C21H23Cl2N2O6P
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:250 mg/mL (498.70 mM; Need ultrasonic)
  • SMILES
    O=P(O)(O)CC1=CC=C(NC(C2CCN(C(OCC3=CC(Cl)=CC(Cl)=C3)=O)CC2)=O)C=C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Balupuri A, et al. Discovery and optimization of ATX inhibitors via modeling, synthesis and biological evaluation. Eur J Med Chem. 2018 Mar 25;148:397-409.
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